The analysis of competitive, uncompetitive and noncompetitive inhibitors of enzymes can now be extended to understand how the activity of membrane receptors are affected by the binding of drugs. Drugs...The analysis of competitive, uncompetitive and noncompetitive inhibitors of enzymes can now be extended to understand how the activity of membrane receptors are affected by the binding of drugs. Drugs targeted to membrane receptors can have a variety of effects. They may elicit the same biological effects as the natural ligand. If so, they are called agonists. Conversely they may inhibit the biological activity of the receptor. If so they called antagonists
In most instances of natural neuron inhibition GABA is the inhibitory transmitter. GABA has the specific effect of opening anion channels in nerves, allowing large numbers of chloride ions to diffuse ...In most instances of natural neuron inhibition GABA is the inhibitory transmitter. GABA has the specific effect of opening anion channels in nerves, allowing large numbers of chloride ions to diffuse into the terminal fibril.
